Dileucine Capsules (2000mg) 50 Count Leucine Dipeptide: Two L-leucine residues (Leu-Leu), 244.33 Da, ≥98% purity PEPT1 Transport System: Active absorption via proton-coupled peptide transporter in small intestine Muscle Protein Synthesis: Enhanced mTORC1 activation and 42% greater anabolic response versus free leucine Manufacturer: RiboCore Availability: In stock SKU: RC-DILEUCINE-CAPSULES-2 $1.00 Qty: Add to cart Ship to Select country United States of America Afghanistan Åland Islands Albania Algeria American Samoa Andorra Angola Anguilla Antarctica Antigua and Barbuda Argentina Armenia Aruba Australia Austria Azerbaijan Bahamas Bahrain Bangladesh Barbados Belarus Belgium Belize Benin Bermuda Bhutan Bolivia (Plurinational State of) Bonaire, Sint Eustatius and Saba Bosnia and Herzegovina Botswana Bouvet Island Brazil British Indian Ocean Territory Brunei Darussalam Bulgaria Burkina Faso Burundi Cabo Verde Cambodia Cameroon Canada Cayman Islands Central African Republic Chad Chile China Christmas Island Cocos (Keeling) Islands Colombia Comoros Congo Congo (Democratic Republic of the) Cook Islands Costa Rica Côte d'Ivoire Croatia Cuba Curaçao Cyprus Czechia Denmark Djibouti Dominica Dominican Republic Ecuador Egypt El Salvador Equatorial Guinea Eritrea Estonia Eswatini Ethiopia Falkland Islands (Malvinas) Faroe Islands Fiji Finland France French Guiana French Polynesia French Southern Territories Gabon Gambia Georgia Germany Ghana Gibraltar Greece Greenland Grenada Guadeloupe Guam Guatemala Guernsey Guinea Guinea-Bissau Guyana Haiti Heard Island and McDonald Islands Holy See Honduras Hong Kong Hungary Iceland India Indonesia Iran (Islamic Republic of) Iraq Ireland Isle of Man Israel Italy Jamaica Japan Jersey Jordan Kazakhstan Kenya Kiribati Korea (Democratic People's Republic of) Korea (Republic of) Kuwait Kyrgyzstan Lao People's Democratic Republic Latvia Lebanon Lesotho Liberia Libya Liechtenstein Lithuania Luxembourg Macao Madagascar Malawi Malaysia Maldives Mali Malta Marshall Islands Martinique Mauritania Mauritius Mayotte Mexico Micronesia (Federated States of) Moldova (Republic of) Monaco Mongolia Montenegro Montserrat Morocco Mozambique Myanmar Namibia Nauru Nepal Netherlands New Caledonia New Zealand Nicaragua Niger Nigeria Niue Norfolk Island North Macedonia Northern Mariana Islands Norway Oman Pakistan Palau Palestine, State of Panama Papua New Guinea Paraguay Peru Philippines Pitcairn Poland Portugal Puerto Rico Qatar Réunion Romania Russian Federation Rwanda Saint Barthélemy Saint Helena, Ascension and Tristan da Cunha Saint Kitts and Nevis Saint Lucia Saint Martin (French part) Saint Pierre and Miquelon Saint Vincent and the Grenadines Samoa San Marino Sao Tome and Principe Saudi Arabia Senegal Serbia Seychelles Sierra Leone Singapore Sint Maarten (Dutch part) Slovakia Slovenia Solomon Islands Somalia South Africa South Georgia and the South Sandwich Islands South Sudan Spain Sri Lanka Sudan Suriname Svalbard and Jan Mayen Sweden Switzerland Syrian Arab Republic Taiwan, Province of China Tajikistan Tanzania, United Republic of Thailand Timor-Leste Togo Tokelau Tonga Trinidad and Tobago Tunisia Turkey Turkmenistan Turks and Caicos Islands Tuvalu Uganda Ukraine United Arab Emirates United Kingdom of Great Britain and Northern Ireland United States Minor Outlying Islands Uruguay Uzbekistan Vanuatu Venezuela (Bolivarian Republic of) Vietnam Virgin Islands (British) Virgin Islands (U.S.) Wallis and Futuna Western Sahara Yemen Zambia Zimbabwe * Other * Shipping Method Name Estimated Delivery Price No shipping options Apply Custom wishlist OK Add to wishlist Add to compare list Email a friend Technical Specifications CharacteristicValue CAS Number3303-31-9 Molecular Weight244.33 Da Purity≥98% by HPLC FormOral capsules (2000 mg per capsule, 50 count) L-Leucyl-L-Leucine (dileucine) is a bioactive dipeptide composed of two leucine amino acid residues linked by a peptide bond. This compound has emerged as a significant advancement in amino acid supplementation research, demonstrating superior absorption kinetics and biological activity compared to free leucine. Research since the early 2020s has produced over 50 peer-reviewed publications examining its effects on muscle protein synthesis, athletic performance, and sarcopenia research. Dileucine is transported intact across the intestinal epithelium via the proton-coupled peptide transporter PEPT1 (SLC15A1), conferring distinct pharmacokinetic advantages. Studies demonstrate that dileucine ingestion delivers 86% more leucine into skeletal muscle compared to equivalent leucine supplementation within 30 minutes of oral administration, resulting in enhanced activation of anabolic signaling cascades and measurable increases in muscle protein synthesis rates in controlled human trials. Key Research Highlights Research AreaKey Finding Muscle Protein Synthesis2 g dileucine increased muscle protein synthesis rates by 42% compared to equivalent leucine in young males (Oikawa et al. 2021) Strength Gains10-week resistance training with dileucine supplementation produced significantly greater leg press 1RM increases versus placebo and free leucine groups (Zhu et al. 2024) Leucine BioavailabilityDileucine delivered 86% more leucine to skeletal muscle tissue within 30 minutes compared to free leucine (Oikawa et al. 2021) Research Applications Muscle protein synthesis and anabolism research Exercise physiology and athletic performance studies Sarcopenia and age-related muscle loss research Intestinal peptide transport and nutrient absorption studies mTOR signaling pathway research Metabolic disease and insulin resistance research Pharmaceutical development and drug delivery research